Krystexxa

(pegloticase)

Provider Summary

Primary Uses

Chronic refractory gout in adults who have failed or cannot tolerate conventional urate-lowering therapy.

Mechanism of Action

Pegylated uricase enzyme converts uric acid to allantoin for renal excretion.

Pre-treatment / Baseline Requirement

Screen for G6PD deficiency prior to starting; baseline serum uric acid; premedication and close monitoring for infusion reactions; discontinue if uric acid rises suggesting loss of response.

Common side effects

Infusion reactions, nausea, bruising, nasopharyngitis.

Serious adverse effects / key risks

Boxed warnings: anaphylaxis and infusion reactions; hemolysis/methemoglobinemia in G6PD deficiency.

Referral requirements

Standard infusion referral form + drug-specific checklist

Krystexxa

Patient & Caregiver Education

What it treats

Chronic refractory gout in adults who have failed or cannot tolerate conventional urate-lowering therapy.

How it works

Pegylated uricase enzyme converts uric acid to allantoin for renal excretion.

Before treatment

Tell your clinician if you have an active infection/fever, are pregnant/planning pregnancy, or have major heart/nerve problems. Depending on the medication, you may need labs or screening tests (e.g., TB/hepatitis) and a vaccine review.

Common side effects

Infusion reactions, nausea, bruising, nasopharyngitis.

Get urgent help for:

Boxed warnings: anaphylaxis and infusion reactions; hemolysis/methemoglobinemia in G6PD deficiency.

On treatment Day:

Plan to stay for monitoring. If you feel dizzy, drowsy, or unwell afterward, do not drive and follow your clinician’s instructions.